5-MeO-DALT
5-MeO-DALT or N,N-di allyl-5-methoxy tryptamine is a psychedelic tryptamine first synthesized by Alexander Shulgin.
Chemistry
The full name of the chemical is N-allyl-N- prop-2-en-1- amine. It is related to the compounds 5-MeO-DPT and DALT.In April 2020, Chadeayne et al. solved the crystal structure of the freebase form of 5-MeO-DALT.
Pharmacology
5-MeO-DALT binds to 5-HT1A, 5-HT1D, 5-HT1E, 5-HT2A, 5-HT2B, 5-HT2C, 5-HT6, α2A, α2B, α2C, H1, κ-opioid, σ1 and σ2 receptors with Ki values lower than 10μM and also acts as a DAT and SERT monoamine reuptake inhibitor.Binding site | pKi ± SEM at binding site |
5-HT1A | 7.70 ± 0.10 |
5-HT1B | 6.13 ± 0.04 |
5-HT1D | 7.00 ± 0.10 |
5-HT1E | 6.30 ± 0.05 |
5-HT2A | 6.66 ± 0.08 |
5-HT2B | 7.23 ± 0.05 |
5-HT2C | 6.34 ± 0.08 |
5-HT5A | 5.48 ± 0.04 |
5-HT6 | 6.81 ± 0.03 |
5-HT7 | 7.05 ± 0.07 |
α2A | 6.67 ± 0.07 |
α2B | 6.14 ± 0.04 |
α2C | 5.83 ± 0.06 |
H1 | 6.30 ± 0.06 |
H3 | 5.77 ± 0.04 |
κOR | 5.95 ± 0.07 |
μOR | < 5.00 |
σ1 | 6.52 ± 0.06 |
σ2 | 6.60 ± 0.05 |
DAT | 5.50 ± 0.20 |
NET | < 5.00 |
SERT | 6.30 ± 0.05 |
The metabolism and cytochrome P450 inhibition of 5-MeO-DALT has been described in scientific literature.